Compile Data Set for Download or QSAR
Found 200 of ic50 data for polymerid = 50000030,50000851,50002755
LigandPNGBDBM83720(6-(2-naphthalenylsulfonyl)quinazoline-2,4-diamine ...)copy SMILEScopy InChI
Affinity DataIC50: 0.0200nMAssay Description:Antibacterial activity against Streptococcus faecalis assessed as growth inhibitionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SWQPubMed
LigandPNGBDBM50614282(CHEMBL5279964)copy SMILES
Affinity DataIC50: 6.90nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50614275(CHEMBL5277226)copy SMILES
Affinity DataIC50: 9.20nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50614276(CHEMBL5286888)copy SMILES
Affinity DataIC50: 9.90nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50614277(CHEMBL5267440)copy SMILES
Affinity DataIC50: 11nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50614279(CHEMBL5279347)copy SMILES
Affinity DataIC50: 11nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50614280(CHEMBL5276161)copy SMILES
Affinity DataIC50: 12nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50614431(CHEMBL5289236)copy SMILES
Affinity DataIC50: 12nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50614274(CHEMBL5272543)copy SMILES
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50614281(CHEMBL5288022)copy SMILES
Affinity DataIC50: 15nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50614278(CHEMBL5285039)copy SMILES
Affinity DataIC50: 16nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50350465(AMPICILLIN | AY-6108 | Amcill | Aminobenzylpenicil...)copy SMILEScopy InChI
Affinity DataIC50: 28.6nMAssay Description:Antibacterial activity against Streptococcus faecalis by broth microdilution techniqueMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6GNNPubMed
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 36.2nMAssay Description:Antibacterial activity against Enterococcus faecalis MTCC 439 incubated overnight by broth dilution techniqueMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7SD8PubMed
LigandPNGBDBM50335519((S)-3,6-Diamino-hexanoic acid {(3S,9S,12S,15S)-3-(...)copy SMILEScopy InChI
Affinity DataIC50: 41.4nMAssay Description:Antibacterial activity against gram positive bacteria Enterococcus faecalis was determined by twofold Micro-broth dilution assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FJ2JZ3PubMed
LigandPNGBDBM50614273(CHEMBL5279536)copy SMILES
Affinity DataIC50: 53nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM50498223(CHEMBL3577359)copy SMILEScopy InChI
Affinity DataIC50: 167nMAssay Description:Antibacterial activity against Enterococcus faecalis ATCC 51299 assessed as growth inhibition using fresh sample in DMSO by CLSI methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5R6XPubMed
LigandPNGBDBM50225960(CHEMBL310176)copy SMILEScopy InChI
Affinity DataIC50: 219nMAssay Description:Concentration (IC50) to inhibit the growth of Streptococcus faecalis.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2X9WPubMed
LigandPNGBDBM50225959(CHEMBL307316)copy SMILEScopy InChI
Affinity DataIC50: 401nMAssay Description:Concentration (IC50) to inhibit the growth of Streptococcus faecalis.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2X9WPubMed
LigandPNGBDBM50476074(Gentamicin | SCH-9724 | Uromycine)copy SMILEScopy InChI
Affinity DataIC50: 445nMAssay Description:Antibacterial activity against Streptococcus faecalis by broth microdilution techniqueMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6GNNPubMed
LigandPNGBDBM50600678(CHEMBL5176174)copy SMILES
Affinity DataIC50: 500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H9997NPubMed
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 603nMAssay Description:Antibacterial activity against Enterococcus faecalis ATCC 51299 assessed as growth inhibition using fresh sample in DMSO by CLSI methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5R6XPubMed
LigandPNGBDBM50366826(DR-3355 | Floxacin | Iquix | LEVOFLOXACIN | Levaqu...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Antibacterial activity against vancomycin-sensitive Enterococcus faecalis 12-5 after 18 hrs by broth microdilution methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2280BKRPubMed
LigandPNGBDBM50366826(DR-3355 | Floxacin | Iquix | LEVOFLOXACIN | Levaqu...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Antibacterial activity against vancomycin-sensitive Enterococcus faecalis ATCC 29212 after 18 hrs by broth microdilution methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2280BKRPubMed
LigandPNGBDBM50509323(CHEMBL4436622)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Antibacterial activity against vancomycin-resistant Enterococcus faecalis AUS-RBWH-VRE-01 assessed as reduction in fungal growth incubated for 24 hrs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5KB8PubMed
LigandPNGBDBM50366826(DR-3355 | Floxacin | Iquix | LEVOFLOXACIN | Levaqu...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Antibacterial activity against vancomycin-resistant Enterococcus faecalis ATCC 51299 after 18 hrs by broth microdilution methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2280BKRPubMed
LigandPNGBDBM31768(CHEMBL295698 | Ketoconazole | Nizoral | Panfungol)copy SMILEScopy InChI
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of cholesterol side chain cleavage cytochrome P450More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7SZTPubMed
LigandPNGBDBM50497194(CHEMBL3116168)copy SMILEScopy InChI
Affinity DataIC50: 1.44E+3nMAssay Description:Antimicrobial activity against Enterococcus faecalis assessed as inhibition of biofilm formation after 20 hrs by crystal violet staining analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4F6VPubMed
LigandPNGBDBM50237605(Achromycin | Achromycin V | CHEBI:27902 | Cyclopar...)copy SMILEScopy InChI
Affinity DataIC50: 1.57E+3nMAssay Description:Antibacterial activity against vancomycin-resistant Enterococcus faecalis ATCC 51299 after 18 hrs by broth dilution assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FNXPubMed
LigandPNGBDBM50509324(CHEMBL4463460)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Antibacterial activity against vancomycin-resistant Enterococcus faecalis AUS-RBWH-VRE-01 assessed as reduction in fungal growth incubated for 24 hrs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5KB8PubMed
LigandPNGBDBM50478886(CHEMBL501116)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Antibacterial activity against vancomycin-resistant Enterococcus faecalis ATCC 51299 after 18 hrs by broth dilution assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FNXPubMed
LigandPNGBDBM50497201(CHEMBL3116167)copy SMILEScopy InChI
Affinity DataIC50: 2.17E+3nMAssay Description:Antimicrobial activity against Enterococcus faecalis assessed as inhibition of biofilm formation after 20 hrs by crystal violet staining analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4F6VPubMed
LigandPNGBDBM50103513(CHEBI:17076 | Chemform | Gerox | NSC-14083 | Strep...)copy SMILEScopy InChI
Affinity DataIC50: 2.23E+3nMAssay Description:Antibacterial activity against gram positive bacteria Enterococcus faecalis was determined by twofold Micro-broth dilution assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FJ2JZ3PubMed
LigandPNGBDBM50499513(CHEMBL4299436)copy SMILEScopy InChI
Affinity DataIC50: 2.27E+3nMAssay Description:Antibacterial activity against low level vancomycin-resistant Enterococcus faecalis ATCC 51299 by plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61P8HPubMed
LigandPNGBDBM50497203(CHEMBL3115985)copy SMILEScopy InChI
Affinity DataIC50: 2.29E+3nMAssay Description:Antimicrobial activity against Enterococcus faecalis assessed as inhibition of biofilm formation after 20 hrs by crystal violet staining analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4F6VPubMed
LigandPNGBDBM50335519((S)-3,6-Diamino-hexanoic acid {(3S,9S,12S,15S)-3-(...)copy SMILEScopy InChI
Affinity DataIC50: 2.34E+3nMAssay Description:Antibacterial activity against Enterococcus faecalis ATCC 51299 assessed as growth inhibition using fresh sample in DMSO by CLSI methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5R6XPubMed
LigandPNGBDBM50497199(CHEMBL3115992)copy SMILEScopy InChI
Affinity DataIC50: 2.38E+3nMAssay Description:Antimicrobial activity against Enterococcus faecalis assessed as inhibition of biofilm formation after 20 hrs by crystal violet staining analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4F6VPubMed
LigandPNGBDBM50497204(CHEMBL3115986)copy SMILEScopy InChI
Affinity DataIC50: 2.39E+3nMAssay Description:Antimicrobial activity against Enterococcus faecalis assessed as inhibition of biofilm formation after 20 hrs by crystal violet staining analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4F6VPubMed
LigandPNGBDBM50218278(CHEMBL279571)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Compound was evaluated for inhibition of peptidoglycan synthesis in Enterococcus faecalis using [14C]lysine radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D79DM6PubMed
LigandPNGBDBM50335519((S)-3,6-Diamino-hexanoic acid {(3S,9S,12S,15S)-3-(...)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Compound was evaluated for inhibition of peptidoglycan synthesis in Enterococcus faecalis using [14C]lysine radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D79DM6PubMed
LigandPNGBDBM50600667(CHEMBL5180164)copy SMILES
Affinity DataIC50: 2.70E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H9997NPubMed
LigandPNGBDBM50498339(CHEMBL3585711)copy SMILEScopy InChI
Affinity DataIC50: 2.72E+3nMAssay Description:Antibacterial activity against Enterococcus faecalis CECT 481 assessed as inhibition of microbial growth incubated for 18 hrs by 2-fold microtiter br...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56NRFPubMed
LigandPNGBDBM50497190(CHEMBL3115993)copy SMILEScopy InChI
Affinity DataIC50: 2.85E+3nMAssay Description:Antimicrobial activity against Enterococcus faecalis assessed as inhibition of biofilm formation after 20 hrs by crystal violet staining analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4F6VPubMed
LigandPNGBDBM50004442((2S,4S)-ketoconazole | 1-acetyl-4-(4-{[(2S,4S)-2-(...)copy SMILEScopy InChI
Affinity DataIC50: 2.95E+3nMAssay Description:Inhibition of cholesterol side chain cleavage cytochrome P450More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7SZTPubMed
LigandPNGBDBM50600670(CHEMBL5204687)copy SMILES
Affinity DataIC50: 3.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H9997NPubMed
LigandPNGBDBM50498341(CHEMBL3585709)copy SMILEScopy InChI
Affinity DataIC50: 3.06E+3nMAssay Description:Antibacterial activity against Enterococcus faecalis CECT 481 assessed as inhibition of microbial growth incubated for 18 hrs by 2-fold microtiter br...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56NRFPubMed
LigandPNGBDBM50600662(CHEMBL5193721)copy SMILES
Affinity DataIC50: 3.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H9997NPubMed
LigandPNGBDBM50497191(CHEMBL3116162)copy SMILEScopy InChI
Affinity DataIC50: 3.14E+3nMAssay Description:Antimicrobial activity against Enterococcus faecalis assessed as inhibition of biofilm formation after 20 hrs by crystal violet staining analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4F6VPubMed
LigandPNGBDBM50498340(CHEMBL3585717)copy SMILEScopy InChI
Affinity DataIC50: 3.19E+3nMAssay Description:Antibacterial activity against Enterococcus faecalis CECT 481 assessed as inhibition of microbial growth incubated for 18 hrs by 2-fold microtiter br...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56NRFPubMed
LigandPNGBDBM50498338(CHEMBL3585716)copy SMILEScopy InChI
Affinity DataIC50: 3.66E+3nMAssay Description:Antibacterial activity against Enterococcus faecalis CECT 481 assessed as inhibition of microbial growth incubated for 18 hrs by 2-fold microtiter br...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56NRFPubMed
LigandPNGBDBM50497202(CHEMBL3115977)copy SMILEScopy InChI
Affinity DataIC50: 3.69E+3nMAssay Description:Antimicrobial activity against Enterococcus faecalis assessed as inhibition of biofilm formation after 20 hrs by crystal violet staining analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4F6VPubMed
Displayed 1 to 50 (of 200 total ) | Next | Last >>
Jump to: